881417-31-8Relevant articles and documents
Efficient synthesis of functionalized benzazepine derivatives utilizing intramolecular mitsunobu reaction
Ohtani, Tadaaki,Kawano, Yoshikazu,Kitano, Kazuyoshi,Matsubara, Jun,Komatsu, Makoto,Uchida, Minoru,Tabusa, Fujio,Nagao, Yoshimitsu
, p. 481 - 502 (2007/10/03)
The 5-hydroxy-2,3,4,5-tetrahydro-1H-benzazepine derivative (2), which is a typical metabolite of mozavaptan (1) having the 2,3,4,5-tetrahydro-1H-benzazepine skeleton, was synthesized by utilizing the intramolecular Mitsunobu reaction of the corresponding