883565-87-5Relevant articles and documents
Synthesis and evaluation of [11C]RU40555, a selective glucocorticoid receptor antagonist
Matsuya, Takahiro,Takamatsu, Hiroyuki,Murakami, Yoshihiro,Noda, Akihiro,Osoda, Kazuhiko,Ichise, Rikiya,Awaga, Yuji,Nishimura, Shintaro
, p. 657 - 668 (2007/10/03)
We demonstrated the synthesis of carbon-11 labeled 17-α-hydroxy-11- β-/4-/[methyl]-[1-methylethyl]-aminophenyl/-17α-[prop-1-ynyl] esta-4-9-diene-3-one (RU40555), a selective glucocorticoid receptor (GR) antagonist, and examined the in vivo profile of [su