88369-83-9Relevant articles and documents
Selective synthesis of 1 -functionalized-alkyl-1H-indazoles
Hunt, Kevin W.,Moreno, David A.,Suiter, Nicole,Clark, Christopher T.,Kim, Ganghyeok
scheme or table, p. 5054 - 5057 (2009/12/28)
An efficient method for the selective "N1" alkylation of indazoles is described. Use of a-halo esters, lactones, ketones, amides, and bromoacetonitrile provides good to excellent yield of the desired N1 products.