88939-68-8Relevant academic research and scientific papers
ZnO-mediated regioselective C-arylsulfonylation of indoles: A facile solvent-free synthesis of 2- and 3-sulfonylindoles and preliminary evaluation of their activity against drug-resistant mutant HIV-1 reverse transcriptases (RTs)
Tocco, Graziella,Begala, Michela,Esposito, Francesca,Caboni, Pierluigi,Cannas, Valeria,Tramontano, Enzo
, p. 6237 - 6241 (2013/10/22)
A ZnO-mediated one-pot solvent-free protocol for the regioselective C-arylsulfonylation of indoles is described and some novel derivatives were tested on wild type and non-nucleoside inhibitor resistant K103N and Y181C HIV-1 reverse transcriptases (RTs).
INDOLE-2,3-QUINODIMETHANES. SYNTHESIS OF INDOLOCARBAZOLES FOR THE SYNTHESIS OF THE FUSED DIMERIC INDOLE ALKALOID STAUROSPORINONE
Magnus, Philip D.,Exon, Christopher,Sear, Nancy L.
, p. 3725 - 3730 (2007/10/02)
N--3-ethyl-2-formylindole, made by direct electrophilic formylation of N--3-ethylindole using α,α-dichloromethylmethylether/TiCl4, was converted into the imine 23 by treatment with 2-aminostyrene.The i
