893602-41-0Relevant academic research and scientific papers
BET-PROTEIN INHIBITING 3,4-DIHYDROPYRIDO[2,3-B]PYRAZINONES WITH META-SUBSTITUTED AROMATIC AMINO- OR ETHER GROUPS
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Paragraph 0871; 0872; 0873, (2017/05/19)
The present invention relates to BET protein-inhibitory, especially BRD4-inhibitory 3,4-dihydropyrido[2,3-b]pyrazinones with a meta-substituted aromatic amino or ether group of the general formula (I) in which A, X, Y, R1, R2, R
A mild and efficient synthesis of aryl sulfones from aryl chlorides and sulfinic acid salts using microwave heating
Yuan, Yan-Qin,Guo, Sheng-Rong
supporting information; experimental part, p. 2750 - 2756 (2011/12/04)
The CuCl-catalyzed coupling of aryl chlorides and sulfinic acid salts provides a simple and extremely efficient route to unsymmetrical aryl sulfones in high to excellent yields under microwave irradiation within 3-30 minutes. Georg Thieme Verlag Stuttgart · New York.
