900512-29-0Relevant academic research and scientific papers
Triazole oxytocin antagonists: Identification of an aryloxyazetidine replacement for a biaryl substituent
Brown, Alan,Brown, T. Bruce,Calabrese, Andrew,Ellis, Dave,Puhalo, Nicholas,Ralph, Michael,Watson, Lesa
scheme or table, p. 516 - 520 (2010/04/05)
A series of aryloxyazetidines, aryloxypyrrolidines and aryloxypiperidines were designed based on structural overlap with previously reported arylpyrazine Oxytocin antagonists. Similarly high levels of Oxytocin antagonism were achievable in these new serie
Substituted triazole derivatives as oxytocin antagonists
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Page/Page column 37-38, (2008/06/13)
The present invention relates to substituted triazoles of formula (I), uses thereof, processes for the preparation thereof and compositions containing said compounds. These inhibitors have utility in a variety of therapeutic areas including sexual dysfunction.
