912848-72-7Relevant academic research and scientific papers
Identification of a manufacturing route of novel CRF-1 antagonists containing a 2,3-Dihydro-1 H-pyrrolo[2,3-b]pyridine moiety
Ribecai, Arianna,Bacchi, Sergio,Delpogetto, Monica,Guelfi, Simone,Manzo, Angelo Maria,Perboni, Alcide,Stabile, Paolo,Westerduin, Pieter,Hourdin, Marie,Rossi, Sara,Provera, Stefano,Turco, Lucilla
experimental part, p. 895 - 901 (2011/03/20)
A case study on the synthesis of novel CRF-1 antagonists containing the 2,3-dihydro-1H-pyrrolo[2,3-b]pyridine moiety is presented. The development of ever more efficient synthetic routes allowed the progression of three candidates at the same time. A manu
PROCESS FOR PREPARING BICYCLIC COMPOUNDS
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Page/Page column 23, (2008/06/13)
The present invention relates to a novel process for preparing compounds of formula (IA), which are potent and specific antagonists of corticotropin-releasing factor (CRF) receptors, from intermediate compounds of formula (I), by a coupling reaction catal
PROCESS FOR PREPARING BICYCLIC COMPOUNDS
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Page/Page column 17-18, (2008/06/13)
The present invention relates to a process for preparing compounds of formula (IA), which are potent and specific antagonists of corticotropin-releasing factor (CRF) receptors, from intermediate compounds of formula (I), by a coupling reaction catalysed b
