913836-10-9

Usage

Uses

Used in Pharmaceutical Industry:
3-Borono-2-methoxybenzoic acid is used as a building block for the synthesis of various pharmaceuticals. Its boronic acid group allows for the formation of reversible covalent bonds with other molecules, which is useful in the development of medicinal drugs.
Used in Agrochemical Industry:
3-Borono-2-methoxybenzoic acid is also used as a building block in the synthesis of agrochemicals. Its versatile structure and properties make it a valuable compound in the development of agricultural chemicals.
Used in Chemical Research:
3-Borono-2-methoxybenzoic acid is utilized in chemical research for its unique properties, such as the ability to form reversible covalent bonds. This makes it a valuable tool in the study of chemical reactions and the development of new chemical compounds.
Used in Drug Development:
3-Borono-2-methoxybenzoic acid is used in drug development due to its potential to enhance the properties of medicinal drugs. Its boronic acid group can form reversible covalent bonds, which can improve the drug's efficacy and selectivity.
Used in Chemical Sensors:
3-Borono-2-methoxybenzoic acid is used in the development of chemical sensors due to its ability to form reversible covalent bonds with other molecules. This property allows for the detection and measurement of specific chemical compounds, making it a valuable component in sensor technology.

InChI:InChI=1/C8H9BO5/c1-14-7-5(8(10)11)3-2-4-6(7)9(12)13/h2-4,12-13H,1H3,(H,10,11)

Upstream product

• 124-38-9 carbon dioxide 
• 38603-09-7 2,6-dibromoanisole 

Downstream Products

• 1256337-30-0 [4-[2-(3-tert-butoxycarbonyl-2-methoxy-phenyl)-1-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl)-ethylcarbamoyl]-benzyl]-triethyl-ammonium bromide 
• 1256336-60-3 [4-[2-(3-tert-butoxycarbonyl-2-methoxy-phenyl)-1-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl)-ethylcarbamoyl]-benzyl]-pyridinium bromide 
• 1256335-63-3 (1R)-(4-(triethylamino)-methyl)-benzoylamino-(3-carboxy-2-hydroxy)benzyl-methyl boronic acid bromide 
• 1256336-76-1 3-(2-(3-((acetyl-(2-tert-butoxycarbonylamino-ethyl)-amino)-methyl)-benzoylamino)-2-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl)-ethyl)-2-methoxy-benzoic acid tert-butyl ester 
• 1256336-56-7 2-methoxy-3-[2-((4-boc-piperazinylmethyl)-benzoylamino)-2-{2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl}-ethyl]-benzoic acid tert-butyl ester 
• 1256337-23-1 3-[2-[(4-(benzyloxycarbonylamino-imino-methyl)-phenyl)acetylamino]-2-(2,9,9-trimethyl-3,5-doxa-4-bora-tricyclo[6.1.1.0.(2,6)]dec-4-yl)-ethyl]-2-methoxy-benzoic acid tert-butyl ester 
• 1256336-62-5 {4-[2-(3-tert-butoxycarbonyl-2-methoxy-phenyl)-1-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6,1,1,0(2,6)]dec-4-yl)-ethylcarbamoyl]-benzyl}-2-tert-butoxycarbonylamino-ethylamine 
• 1256336-59-0 1-{4-[2-(3-tert-butoxycarbonyl-2-methoxy-phenyl)-1-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl)-ethyl-carbamoyl]benzyl}piperidine-3-caroxylic acid ethyl ester 
• 1256336-66-9 3-[2-{3-((2-tert-butoxycarbonylamino-ethylamino)-methyl)-benzoylamipo}-2-(2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0(2,6)]dec-4-yl)-ethyl]-2-methoxy-benzoic acid tert-butyl ester 
• 1256336-61-4 (1R)-[4-(pyridinium)-methyl]-benzoylamino-(3-carboxy-2-hydroxy)benzyl-methyl boronic acid chloride 
• 1256337-19-5 3-[2-(2-(4-((tert-butoxycarbonylmethyl)-aminomethyl)-phenyl)-acetylamino)-2-(2,9,9-trimethyl-3,5-doxa-4-bora-tricyclo[6.1.1.0.(2,6)]dec-4-yl)-ethyl]-2-methoxy-benzoic acid tert-butyl ester 

Relevant academic research and scientific papers

One-pot generation of lithium (lithiophenyl)trialkoxyborates from substituted dihalobenzenes (Hal = Br, I) and their derivatization with electrophiles

The simple one-pot approach to synthetically useful phenyltrialkoxyborates bearing lithium at the phenyl ring has been developed starting with 1,3- and 1,4-diiodobenzene, as well as several activated dibromobenzenes and bromoiodobenzenes. The general sequence of transformations involves halogen-lithium exchange by using nBuLi and subsequent boronation with a trialkylborate. The resulting lithium (halophenyl) trialkoxyborates were then subjected to halogen-lithium exchange in situ with a second equivalent of nBuLi to give dianionic lithium (lithiophenyl)trialkoxyborates. Treatment with selected electrophiles afforded substituted arylboronic acids and/or their pinacol esters as final products in moderate-to-good yields. Wiley-VCH Verlag GmbH & Co. KGaA, 2008.