914200-90-1Relevant articles and documents
QUINOLINE DERIVATIVES AS KINASE ENZYME INHIBITORS
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, (2010/11/24)
Compounds of formula (IA) or (IB) are inhibitors of aurora kinase activity, and are useful in the treatment of cell proliferation disease and other conditions associated with inappropriate aurora kinase activity wherein R1 is a carboxylic acid
ENZYME AND RECEPTOR MODULATION
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Page/Page column 56, (2008/06/13)
Covalent conjugation of an alpha amino acid ester to a modulator of the activity of a target intracellular enzyme or receptor, wherein the ester group of the conjugate is hydrolysable by one or more intracellular carboxylesterase enzymes to the correspond