915407-79-3Relevant academic research and scientific papers
Tricyclic HIV integrase inhibitors: Potent and orally bioavailable C5-aza analogs
Jin, Haolun,Wright, Matthew,Pastor, Richard,Mish, Michael,Metobo, Sammy,Jabri, Salman,Lansdown, Rachael,Cai, Ruby,Pyun, Peter,Tsiang, Manuel,Chen, Xiaowu,Kim, Choung U.
, p. 1388 - 1391 (2008/09/19)
A series of C5-aza tricyclic HIV integrase inhibitors was prepared. A highly potent and orally bioavailable compound (compound 9) was identified and selected for development.
Integrase inhibitor compounds
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Page/Page column 65, (2010/11/26)
Tricyclic compounds, protected intermediates thereof, and methods for inhibition of HIV-integrase are disclosed.
