915943-50-9Relevant academic research and scientific papers
A concise synthesis of 5-demethyl-HKI 0231A and 5-demethyl-HKI 0231B
Kraus, George A.,Wu, Tao
, p. 7801 - 7803 (2006)
The pentacyclic skeleton of HKI 0231A and HKI 0231B was synthesized by a novel radical cyclization/oxidation followed by DDQ oxidation to introduce the methoxyl groups. This is the first synthetic pathway to both the HKI 0231A and the HKI 0231B series.
