920012-15-3Relevant articles and documents
Synthesis of biotinylated photoaffinity probes based on arylsulfonamide γ-secretase inhibitors
Fuwa, Haruhiko,Hiromoto, Kenichi,Takahashi, Yasuko,Yokoshima, Satoshi,Kan, Toshiyuki,Fukuyama, Tohru,Iwatsubo, Takeshi,Tomita, Taisuke,Natsugari, Hideaki
, p. 4184 - 4189 (2007/10/03)
Synthesis and biological evaluation of an arylsulfonamide class of γ-secretase inhibitors are described. Design, synthesis, and biological evaluation of multifunctional molecular probes harboring a benzophenone photophore as a cross-linking group and a biotin tag are also reported.