929804-33-1Relevant academic research and scientific papers
NEW DERIVATIVES OF INDOLE FOR THE TREATMENT OF CANCER, VIRAL INFECTIONS AND LUNG DISEASES
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Page/Page column 52, (2014/06/24)
The present invention relates to a new class of indole derivatives, having a particular MKlp2 inhibition profile and useful as a therapeutic agent, in particular for the treatment of cancer, viral infections and lung diseases.
NOVEL SMALL MOLECULE POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS I
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Page/Page column 26, (2011/10/13)
The present invention relates to small molecule potentiators of metabotropic receptors, in particular of the mGlu2 receptor. The present invention also relates to the use of these compounds for the prevention or treatment of neurological and psychiatric d
Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockers
Knutsen, Lars J.S.,Hobbs, Christopher J.,Earnshaw, Christopher G.,Fiumana, Andrea,Gilbert, Jenny,Mellor, Sarah L.,Radford, Fleur,Smith, Nichola J.,Birch, Philip J.,Russell Burley,Ward, Stuart D.C.,James, Iain F.
, p. 662 - 667 (2007/10/03)
A series of new N-type (Cav2.2) calcium channel blockers derived from the 'hit' structures 2-(3-bromo-4-fluorophenyl)-3-(2-pyridin-2-ylethyl)thiazolidin-4-one 9 and its 2-[4-(4-bromophenyl)pyridin-3-yl]-3-isobutyl analogue 10 is described. Exte
