930587-03-4

Upstream product

• 930587-02-3 (4S,1'S)-4-[1'-(2''-benzyloxy-ethyl)-allyl]-2,2-dimethyl-oxazolidine-3-carboxylic acid tert-butyl ester 
• 100-39-0 benzyl bromide 
• 515173-88-3 (1'S,4S)-4-[1'-(2''-hydroxy-ethyl)-allyl]-2,2-dimethyl-oxazolidine-3-carboxylic acid tert-butyl ester 

Downstream Products

• 930587-04-5 (S)-4-[(S)-1-(2-Benzyloxy-ethyl)-3-methanesulfonyloxy-propyl]-2,2-dimethyl-oxazolidine-3-carboxylic acid tert-butyl ester 
• 930587-05-6 (2S,3R)-3-(2'-benzyloxy-ethyl)-pyrrolidine-1,2-dicarboxylic acid 1-tert-butyl ester 2-methyl ester 

Relevant academic research and scientific papers

Synthesis of conformationally constrained analogues of RGD tripeptide

Convergent syntheses of N-functionalized (3S,4S)-3-amino-4-vinyl-piperidin-2-one 10, trans-3-substituted proline 18 and (3S)-3-amino-piperidin-2-one 28 are developed. By incorporating these building blocks to an appropriate position, conformationally cons