935248-22-9Relevant academic research and scientific papers
A novel, non-substrate-based series of glycine type 1 transporter inhibitors derived from high-throughput screening
Lowe,Drozda,Qian,Peakman,Liu,Gibbs,Harms,Schmidt,Fisher,Strick,Schmidt,Vanase,Lebel
, p. 1675 - 1678 (2007/10/03)
The synthesis and structure-activity relationships (SAR) of a series of indane and tetralin inhibitors of the type 1 glycine transporter, derived from a high-throughput screening (HTS) hit, are described. Key modifications that reduced the 5HT1B receptor
