93591-79-8

Upstream product

• 93591-78-7 1-[4-(2-benzoylphenylamino)piperidin-1-yl]ethanone 
• 93593-07-8 2-benzoyl-N-(1-methyl-4-piperidinyl)aniline 
• 93592-27-9 2-benzoyl-N-(4-piperidinyl)aniline 
• 93592-26-8 N-<1-(ethoxycarbonyl)-4-piperidinyl>-2-benzoylaniline 

Relevant academic research and scientific papers

1-Azacycloalkyl-1,4-benzodiazepin-2-ones with Antianxiety-Antidepressant Actions

A series of 1-azacycloalkyl-1,4-benzodiazepin-2-ones were synthesized from 1-azacycloalkyl-2-benzoylanilines 2-4 and corresponding imines 5 and 6 and then evaluated for their central nervous system activities.Pharmacological data showed that some of these

1,4-Benzodiazepine derivatives

1,4-Benzodiazepine derivatives of the formula: STR1 (in which R1 is pyrrolidinyl or piperidinyl each optionally substituted by C1-3 alkyl, phenyl-C1-3 alkyl, C1-5 alkanoyl, or C2-5 alkoxycarbonyl, R2 is hydrogen, hydroxy, or acetoxy, R3 is C1-3 alkyl, phenyl-C1-3 alkyl, or phenyl optionally substituted by one or two halogens, X is hydrogen, halogen, C1-3 alkyl, C1-3 alkoxy, nitro, trifluoromethyl, or di-C1-3 alkyl-amino, and n is 1 or 2) or pharmaceutically acceptable acid addition salts thereof, which are useful as a psychotropic agent such as anti-depressant or anxiolytic agent can be prepared from several routes.