949459-68-1Relevant academic research and scientific papers
Synthesis and initial pharmacology of dual-targeting ligands for putative complexes of integrin αvβ3 and PAR2
Dockendorff, Chris,Gandhi, Disha M.,Hernandez, Irene,Holyst, Trudy,Majewski, Mark W.,Rosas, Ricardo,Wang, Zhengli,Weiler, Hartmut,Zhu, Jieqing
, p. 940 - 949 (2020/09/21)
Unpublished data from our labs led us to hypothesize that activated protein C (aPC) may initiate an anti-inflammatory signal in endothelial cells by modulating both the integrin αVβ3 and protease-activated receptor 2 (PAR2), which may exist in close proxi
Peptide backbone modifications on the C-terminal hexapeptide of neurotensin
Einsiedel, Juergen,Huebner, Harald,Hervet, Maud,Haerterich, Steffen,Koschatzky, Susanne,Gmeiner, Peter
, p. 2013 - 2018 (2008/12/22)
To compare backbone-induced susceptibilities with affinity changes that are caused by side-chain modifications in the respective positions, structure activity relationship studies on a series of NT(8-13) analogues were performed providing valuable insight
