95264-91-8

Upstream product

• 118162-45-1 11-azidoundecanoic acid 
• 88313-91-1 6-Amino-hexanethioic acid S-phenyl ester 
• 118162-54-2 11-Azido-undecanethioic acid S-pyridin-2-yl ester 
• 118162-53-1 11-Azido-undecanethioic acid S-phenyl ester 

Relevant academic research and scientific papers

Alternative Procedures for the Macrolactamisation of ω-Azido Acids

ω-Azido acids, after activation of the carboxyl groups as mixed anhydrides, N3(CH2)nCOOCOAr (Ar = 3,5-dinitrophenyl or 2,4,6-trichlorophenyl), can be converted to macrolactams in good yields by treatment with Bu3P under high-dilution conditions; the prese

From Azido Acids to Macrolactams and Macrolactones

A new method is reported for the conversion of azido acids into lactams, via thioester formation and in situ azide reduction and cyclisation under high-dilution conditions; since the quantitative conversion of macrolactams to macrolactones has been shown to be feasible, this results in an indirect, alternative macrolactonisation procedure.