95271-93-5Relevant academic research and scientific papers
Azole endothelin antagonists. 1. A receptor model explains an unusual structure-activity profile
Von Geldern, Thomas W.,Hutchins, Charles,Kester, Jeffrey A.,Wu-Wong, Jinshyun R.,Chiou, William,Dixon, Douglas B.,Opgenorth, Terry J.
, p. 957 - 967 (1996)
The pseudotetrapeptide FR-139317 is a potent and highly selective antagonist of the endothelin-A (ET(A)) receptor; however, its peptidic nature leads to poor oral absorption characteristics which make it an unlikely drug candidate. In an attempt to improv
CALPAIN MODULATORS AND THERAPEUTIC USES THEREOF
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Paragraph 1592, (2018/04/17)
Disclosed herein are small molecule calpain modulator compositions, pharmaceutical compositions, the use and preparation thereof.
