955359-97-4Relevant academic research and scientific papers
The discovery of quinoline based single-ligand human H1and H3receptor antagonists
Procopiou, Panayiotis A.,Ancliff, Rachael A.,Gore, Paul M.,Hancock, Ashley P.,Hodgson, Simon T.,Holmes, Duncan S.,Keeling, Steven P.,Looker, Brian E.,Parr, Nigel A.,Rowedder, James E.,Slack, Robert J.
, p. 5855 - 5859 (2016/12/06)
A novel series of potent quinoline-based human H1and H3bivalent histamine receptor antagonists, suitable for intranasal administration for the potential treatment of allergic rhinitis associated nasal congestion, were identified. Com
QU1NOLINE DERIVATIVES AND THEIR USES FOR RHINITIS AND URTICARIA
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Page/Page column 52-53, (2010/09/17)
The present invention relates to compounds of formula (I) and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various diseases, such as allergic rhinitis.
2-SUBSTITUTED 4-BENZYLPHTHALAZINONE DERIVATIVES AS HISTAMINE H1 AND H3 ANTAGONISTS
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, (2008/06/13)
The present invention relates to compounds of formula (I), and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various disorders, such as allergic rhinitis.
HISTAMINE RECEPTOR ANTAGONISTS COMPRISING AN AZEPIN CORE
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, (2008/06/13)
The present invention relates to compounds of formula (I), and salts thereof, processes for their preparation, to compositions containing them and to their use in the treatment of various disorders, such as allergic rhinitis.
