97457-66-4Relevant academic research and scientific papers
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
Guglielmi, Paolo,Secci, Daniela,Petzer, Anél,Bagetta, Donatella,Chimenti, Paola,Rotondi, Giulia,Ferrante, Claudio,Recinella, Lucia,Leone, Sheila,Alcaro, Stefano,Zengin, Gokhan,Petzer, Jacobus P.,Ortuso, Francesco,Carradori, Simone
, p. 1511 - 1525 (2019/08/26)
A series of benzo[b]thiophen-3-ols were synthesised and investigated as potential human monoamine oxidase (hMAO) inhibitors in vitro as well as ex vivo in rat cortex synaptosomes by means of evaluation of 3,4-dihydroxyphenylacetic acid/dopamine (DOPAC/DA)
Use of Phenacyl Thiosalicylates for the Preparation of 3-Hydroxybenzo[ b ]thiophene Derivatives
Trapani, Patricia,Kvapil, Lubomír,Hradil, Pavel,Soural, Miroslav
supporting information, p. 810 - 814 (2018/02/16)
In this work, we attempted to synthesize thioflavonols using rearrangement of phenacyl thiosalicylates prepared by two different approaches and subjected to cyclization under acidic conditions. Contrary to our expectations, the isolated products were iden
Facile synthesis of 2-substituted benzo[b]thiophen-3-ols in water
Pan, Ben,Ren, Peng,Song, Haibin,Wang, Zhihong
supporting information, p. 1337 - 1344 (2013/05/09)
A facile synthesis of 2-substituted benzo[b]thiophen-3-ols in a simple reaction system is reported with water as the only media. Density functional theory (DFT) investigations suggest two pathways comparable in energetics: A neutral pathway with concerted
Activities of 2-carboxanilido 3-hydroxybenzo[b]thiophens against molluscs Biomphalaria
Gayral,Buisson,Royer
, p. 187 - 189 (2007/10/02)
The title compounds are shown to be nearly as active against molluscs as Niclosamide when they are either dihalogenated or monohalogenated and mononitrated on the benzene ring.
