99347-01-0Relevant articles and documents
Synthesis, structural properties, and pharmacological evaluation of 2-(acylamino)thiophene-3-carboxamides and analogues thereof
Mugnaini, Claudia,Pedani, Valentina,Giunta, Daniela,Sechi, Barbara,Solinas, Maurizio,Casti, Alberto,Castelli, Maria Paola,Giorgi, Gianluca,Corelli, Federico
, p. 1782 - 1793 (2014/01/06)
We have previously reported the synthesis and the pharmacological characterization of a family of methyl 2-(acylamino)thiophene-3-carboxylates as GABAB positive allosteric modulators active both in vitro and in vivo. In the present work, we des
STUDIES ON THE SYNTHESIS OF HETEROCYCLIC COMPOUNDS. PART XII. PYRAZOLO-1,5-BENZODIAZOCINE-4,10-DIONE. A NEW RING SYSTEM
Plescia, Salvatore,Bajardi, Maria Luisa,Daidone, Giuseppe,Roccaro, Angela
, p. 105 - 112 (2007/10/02)
Treatment of N-(1-R-4-carboxypyrazol-5-yl)-2-aminobenzamides 2b,e with thionyl chloride afforded new pyrazolo-1,3-oxazinones 3b,e.When the amide group of compounds 2b,e was blocked pyrazolo-1,5-benzodiazocine-4,10-diones 6a,d were obtained.
Heterocyclic β-Enamino Esters, 39. - Synthesis of 1H-Pyrazolopyrimidines
Wamhoff, Heinrich,Ertas, Muemtaz,Atta, Sanaa M. S.
, p. 1910 - 1916 (2007/10/02)
Die Pyrazol-Enaminoester 1a, b und 4-Pyrazolcarbohydrazide 4a, b sind nuetzliche Ausgangsverbindungen fuer die Darstellung von 1H-Pyrazolopyrimidinen.So ergeben Orthoameisensaeure- und Orthoessigsaeure-triethylester mit 4a, b die 5-(Ethoxymethylena