161609-80-9Relevant articles and documents
TBSOTf-promoted versatile N-formylation using DMF at room temperature
Sakurai, Masayoshi,Kawakami, Rina,Kihara, Nobuhiro
supporting information, p. 1291 - 1294 (2019/04/10)
Hydrazides and amines were N-formylated by DMF in the presence of tert-butyldimethylsilyl triflate (TBSOTf) at room temperature, in good to excellent yields.
AZAINDAZOLES TO TREAT FLAVIVIRIDAE VIRUS INFECTION
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Page/Page column 138; 139, (2011/05/06)
Azaindazole compounds are useful for treating Flaviviridae virus infection, including HCV infection.
Aryl substituted heterocycles
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, (2008/06/13)
The present invention concerns the novel use of aryl substituted heterocycles of formula I, set out below, which antagonize the pharmacological actions of one of ent endogenous neuropeptide tachykinins an the neurokinin 2 (NK2) receptor making them useful whenever such antagonism is desired, such as in the treatment of asthma and related conditions. The invention also provides pharmaceutical compositions containing the aryl substituted heterocycles for use in such treatment. Certain novel aryl substituted heterocycles of formula I and novel intermediates for their manufacture are also provided. STR1