116547-91-2

Basic information

• Product Name: N-(2-Bromophenyl)methansulfonamide
• Synonyms: N-(2-Bromophenyl)methansulfonamide;Methanesulfonamide, N-(2-bromophenyl)-
• CAS NO: 116547-91-2
• Molecular Formula: C₇H₈BrNO₂S
• Molecular Weight: 250.11
• Product Categories: Aryl;Organohalides
• Mol File: 116547-91-2.mol

Chemical Properties

• Appearance: /
• CAS DataBase Reference: N-(2-Bromophenyl)methansulfonamide(CAS DataBase Reference)
• NIST Chemistry Reference: N-(2-Bromophenyl)methansulfonamide(116547-91-2)
• EPA Substance Registry System: N-(2-Bromophenyl)methansulfonamide(116547-91-2)

Safety Data

• Hazardous Substances Data: 116547-91-2(Hazardous Substances Data)

Usage

Uses

Used in Pharmaceutical Synthesis:
N-(2-Bromophenyl)methansulfonamide is used as a key intermediate in the synthesis of pharmaceuticals for its unique chemical properties and reactivity. It serves as a building block in the development of new drugs, particularly in the fields of antibiotics and antifungal agents.
Used in Agrochemical Synthesis:
In the agrochemical industry, N-(2-Bromophenyl)methansulfonamide is utilized as a precursor in the production of various agrochemicals. Its unique chemical properties make it suitable for the development of new compounds with potential applications in agriculture, such as pesticides and herbicides.
Used in Medicinal Chemistry Research:
N-(2-Bromophenyl)methansulfonamide is employed as a research tool in medicinal chemistry. Its unique chemical properties and reactivity make it a valuable compound for exploring new drug candidates and understanding the mechanisms of action in various diseases.
Used in Scientific and Industrial Applications:
Due to its unique chemical properties, N-(2-Bromophenyl)methansulfonamide has potential applications in various scientific and industrial fields. The bromine atom attached to the phenyl ring makes it useful for a wide range of applications, including the development of new materials, catalysts, and chemical processes.

Upstream product

• 124-63-0 methanesulfonyl chloride 
• 615-36-1 2-bromoaniline 

Downstream Products

• 116548-00-6 N-<2-(Trimethylsilylethynyl)phenyl>methanesulfonamide 
• 1206901-63-4 N-(but-2-enyl)-N-(2-bromophenyl)-methanesulfonamide 
• 1206901-65-6 N-(2-bromophenyl)-N-(cyclohex-2-enyl)methanesulfonamide 
• 1206901-64-5 N-(2-bromophenyl)-N-(3-methylbut-2-enyl)methanesulfonamide 
• 1242046-87-2 1-(p-tolyl)quinoxalin-2(1H)-one 
• 553652-34-9 N-(2-bromophenyl)-N-methylmethanesulfonamide 
• 1372589-60-0 N-(2-bromophenyl)-N-ethylmethanesulfonamide 
• 1587691-90-4 N-(2-bromophenyl)-N-(prop-2-ynyl)methanesulfonamide 
• 24827-66-5 1-methyl-1,3-dihydrobenzo[c]isothiazole-2,2-dioxide 

Relevant articles and documents

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The reaction of N-(2-bromophenyl)- and N-(2-iodophenyl)methanesulfonamide with terminal acetylenes in the presence of dichlorobis(triphenylphosphine)palladium yielded 1-methylsulfonylindoles having carbon-functional groups at the 2-position, such as hydroxymethyl, 2-hydroxyethyl, diethoxymethyl, 2-ethoxycarbonylethyl, etc., in one step.Keywords - palladium-catalyzed reaction; dichlorobis(triphenylphosphine)palladium; N-(2-halophenyl)methanesulfonamide; acetylene; 2-substituted 1-methylsulfonylindole.