The fluorine-iminium ion gauche effect: proof of principle and application to asymmetric organocatalysis
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Sparr, Christof,Schweizer, W. Bernd,Senn, Hans Martin,Gilmour, Ryan
supporting information; experimental part
p. 3065 - 3068
(2009/10/01)
4-[6-(2-Aminoethyl)naphthalen-2-yl]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetration
4-[6-(2-Tertiaryaminoethyl)naphthalen-2-yl]benzonitriles are conformationally constrained histamine H3 receptor antagonists with high potency and selectivity. The analogs were designed around a naphthalene core, with the goal of enhancing lipop
Black, Lawrence A.,Nersesian, Diana L.,Sharma, Padam,Ku, Yi-Yin,Bennani, Youssef L.,Marsh, Kennan C.,Miller, Thomas R.,Esbenshade, Timothy A.,Hancock, Arthur A.,Cowart, Marlon
p. 1443 - 1446
(2007/10/03)
Novel amines as histamine-3 receptor ligands and their therapeutic applications
Compounds of formula (I) or a pharmaceutically acceptable salts or prodrug thereof which are useful for the modulation of the histamine-3 receptors in mammals and which are useful for the treatment of disorders ameliorated by histamine-3 receptor ligands.
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(2008/06/13)
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