90226-87-2 Usage
Uses
Used in Cancer Therapy:
CHEMBRDG-BB 4010868 is used as a potential therapeutic agent for cancer treatment. Its inhibitory activity against KDM4 and other histone demethylases can modulate epigenetic regulation, which is often disrupted in cancer cells, leading to uncontrolled cell growth and proliferation. By targeting these enzymes, CHEMBRDG-BB 4010868 may help restore normal epigenetic patterns and inhibit tumor development.
Used in Epigenetics Research:
CHEMBRDG-BB 4010868 is used as a valuable tool in studying epigenetic regulation. Its ability to inhibit KDM4 and other histone demethylases allows researchers to investigate the role of these enzymes in gene expression, cellular differentiation, and disease development. CHEMBRDG-BB 4010868 can help advance our understanding of the complex interplay between genetics and environmental factors in various diseases, including cancer.
Used in Drug Development:
CHEMBRDG-BB 4010868 is used as a lead compound in the development of new drugs targeting histone demethylases. Its inhibitory activity and unique structural features make it a promising starting point for the design and synthesis of more potent and selective inhibitors. These new compounds may offer improved therapeutic efficacy and reduced side effects compared to existing treatments, ultimately benefiting patients with cancer and other diseases associated with epigenetic dysregulation.
Used in Drug Screening and High-Throughput Assays:
CHEMBRDG-BB 4010868 is used as a reference compound in drug screening and high-throughput assays aimed at identifying novel inhibitors of histone demethylases. Its known inhibitory activity serves as a benchmark for evaluating the potency and selectivity of newly synthesized compounds, facilitating the discovery of more effective and safer drugs for cancer therapy and other applications.
Check Digit Verification of cas no
The CAS Registry Mumber 90226-87-2 includes 8 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 5 digits, 9,0,2,2 and 6 respectively; the second part has 2 digits, 8 and 7 respectively.
Calculate Digit Verification of CAS Registry Number 90226-87:
(7*9)+(6*0)+(5*2)+(4*2)+(3*6)+(2*8)+(1*7)=122
122 % 10 = 2
So 90226-87-2 is a valid CAS Registry Number.
InChI:InChI=1/C8H17NO/c1-2-9-5-3-8(7-10)4-6-9/h8,10H,2-7H2,1H3
90226-87-2Relevant articles and documents
COMPOUNDS AND THERAPEUTIC USES THEREOF
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Page/Page column 109, (2010/11/03)
The invention relates to compounds, pharmaceutical compositions, and uses thereof, including therapeutic uses thereof, such as methods useful for treating cancer.
