Orally active esters of dihydroartemisinin: Synthesis and antimalarial activity against multidrug-resistant Plasmodium yoelii in mice

DOI: 10.1016/j.bmcl.2007.12.074

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1436 - 1441 (2008)

Update date:2022-08-04

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Authors:

Singh, Chandan

Chaudhary, Sandeep

Puri, Sunil K.

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Article abstract of DOI:10.1016/j.bmcl.2007.12.074

A series of artemisinin derived esters 7a-j, incorporating pharmacologically privileged substructure, such as biphenyl, adamantane and fluorene, have been prepared and evaluated for antimalarial activity against multidrug-resistant (MDR) Plasmodium yoelii

Full text of DOI:10.1016/j.bmcl.2007.12.074

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