2-[[[2-(2,6-Dimethoxyphenoxy)ethyl]amino]methyl]-1,4-benzoxathian: A new antagonist with high potency and selectivity toward α1-adrenoreceptors

Article abstract of DOI:10.1021/jm00378a001

Much evidence supports the view that the α-adrenoreceptor is not a homogeneous entity. In addition to the classical postsynaptic α-adrenoreceptor, called α₁, that initiates the response of the effector organ, there is a presynaptic α-adrenorece