
Journal of Medicinal Chemistry p. 2724 - 2732 (2009)
Update date:2022-09-26
Topics:
Marco-Contelles, José
León, Rafael
De Los Ríos, Cristóbal
Samadi, Abdelouahid
Bartolini, Manuela
Andrisano, Vincenza
Huertas, Oscar
Barril, Xavier
Luque, F. Javier
Rodríguez-Franco, María I.
López, Beatriz
López, Manuela G.
García, Antonio G.
Carreiras, María Do Carmo
Villarroya, Mercedes
Tacripyrines (1-14) have been designed by combining an AChE inhibitor (tacrine) with a calcium antagonist such as nimodipine and are targeted to develop a multitarget therapeutic strategy to confront AD. Tacripyrines are selective and potent AChE inhibito
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