Bioorganic and Medicinal Chemistry p. 2229 - 2250 (2018)
Update date:2022-08-02
Topics:
Kojima, Takuto
Mochizuki, Michiyo
Takai, Takafumi
Hoashi, Yasutaka
Morimoto, Sachie
Seto, Masaki
Nakamura, Minoru
Kobayashi, Katsumi
Sako, Yuu
Tanaka, Maiko
Kanzaki, Naoyuki
Kosugi, Yohei
Yano, Takahiko
Aso, Kazuyoshi
A new class of corticotropin releasing factor 1 (CRF1) receptor antagonists characterized by a tricyclic core ring was designed and synthesized. Novel tricyclic derivatives 2a–e were designed as CRF1 receptor antagonists based on con
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