Beyond the chiral pool: A general approach to β-amino-α-keto amides

DOI: 10.1016/j.tet.2010.11.018

Source and publish data:

Tetrahedron p. 41 - 47 (2011)

Update date:2022-08-02

Topics:

Authors:

Harrison, Cristian L.

Krawiec, Mariusz

Forslund, Raymond E.

Nugent, William A.

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Article abstract of DOI:10.1016/j.tet.2010.11.018

A simple route was developed for the synthesis of optically enriched β-amino-α-keto amides. The highly diastereoselective addition of alkyl dithiolanecarboxylates to optically enriched sulfinimines affords the corresponding β-amino-α-keto esters in which

Full text of DOI:10.1016/j.tet.2010.11.018

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