Tetrahedron Letters p. 6473 - 6476 (1989)
Update date:2022-07-29
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An in situ production of C-13 acetyl chloride and subsequent reaction with amidrazones affords anxiolytic 1,2,4-triazolobenzodiazepines in reaction times suitable for labelling with carbon-11 (t( 1/2 ) = 20.4 min).
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