Preparation of Nε-(3-hydroxy-16-oxoestra-1,3,5(10)-trien-17β-yl)-L-lysine, 16α-hydroxyesterone-lysine adduct, via Heyns rearrangement

DOI: 10.1016/S0040-4039(00)92047-1

Source and publish data:

Tetrahedron Letters p. 1213 - 1214 (1991)

Update date:2022-08-03

Topics:

Authors:

Miyairi Miyairi

Ichikawa

Nambara Nambara

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)92047-1

Preparation of a stable covalent adduct from 16α-hydroxyestrone with the ε-amino group of lysine via two step reactions involving Schiff base formation followed by Heyns rearrangement is described.

Full text of DOI:10.1016/S0040-4039(00)92047-1

Products guided by the article

Product name:2-tert-Butoxycarbonylamino-6-((8R,9S,13S,14S,17R)-3-hydroxy-13-methyl-16-oxo-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-ylamino)-hexanoic acid

Cas No:133546-19-7

R&D Labs maybe for 133546-19-7

Beijing Harmony Chemical Co., Ltd.

Contact:86-010-84956928

Address:Room 207, Jin feng he B building, No 8 Xin Jie Kou Wai Street, Xi Cheng District, Beijing,PRC. 10008
Xinchang Yueding Chemical Co., Ltd.

Contact:86-571-56926323

Address:NO.90 BEIMENCHENGWAI CHENGGUAN TOWN XINCHANG
KAIYUAN CHEMICAL COMPANY LIMITED.

website:http://www.kaiyuanchem.com

Contact:+86-22-59891255/66/77

Address:B-2205, Kuangshi International Building, Yingbin Road, XiangLuo Bay Business District, Binhai New area, Tianjin, China.
SuZhou LaiTeou

Contact:+86-0512-88957371

Address:shanghai
Henan zhongda Biological Engineering Co., Ltd

Contact:86-28-18109029985

Address:shenzhou road,xuedian industrial estate,zhengzhou city,henan province CHN

Relevant to this article

Photocatalyzed ortho-Alkylation of Pyridine N-Oxides through Alkene Cleavage

Doi:10.1002/anie.201801305
(2018)
Coordination chemistry of the tetraphenyldithioimidodiphosphinate ligand [Ph₂P(S)NP(S)Ph₂]^? and Ph₂P(CH₂)_nPPh₂, n?=?1, 2, 3 toward ReBr(CO)₅

Doi:10.1016/j.ica.2018.12.024
(2019)
A rapid tandem knoevenagel/michael reaction using mohr's salt as a highly efficient catalyst: Green synthesis of bis(pyrazolyl)methanes

Doi:10.2174/1570178612666141204224826
(2015)
Enantioselective epoxidation of unfunctionalized olefins using chiral (salen)manganese(III) complexes

Doi:10.1016/S0040-4039(00)74486-8
(1991)
Synthesis of sequentially deuterated 1-n-Butyl-3-methylimidazolium ionic liquids

Doi:10.1002/jlcr.1884
(2011)
Optically pure bulky (hetero)arylalkyl carbinols via kinetic resolution

Doi:10.1039/c1cc14591f
(2011)

Article Doi