Preparation of Nε-(3-hydroxy-16-oxoestra-1,3,5(10)-trien-17β-yl)-L-lysine, 16α-hydroxyesterone-lysine adduct, via Heyns rearrangement

DOI: 10.1016/S0040-4039(00)92047-1

Source and publish data:

Tetrahedron Letters p. 1213 - 1214 (1991)

Update date:2022-08-03

Topics:

Authors:

Miyairi Miyairi

Ichikawa

Nambara Nambara

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)92047-1

Preparation of a stable covalent adduct from 16α-hydroxyestrone with the ε-amino group of lysine via two step reactions involving Schiff base formation followed by Heyns rearrangement is described.

Full text of DOI:10.1016/S0040-4039(00)92047-1

Products guided by the article

Product name:2-tert-Butoxycarbonylamino-6-((8R,9S,13S,14S,17R)-3-hydroxy-13-methyl-16-oxo-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-ylamino)-hexanoic acid

Cas No:133546-19-7

R&D Labs maybe for 133546-19-7

Chengdu ZY Biochemical Technology Co., LTD

Contact:0086-28-88680086

Address:170 Qingpu Road, Shouan Town, Pujiang County
shandong zhongke taidou chemical co.,ltd

Contact:86-531-88682301

Address:Jinan shandong Province CHina
SHIJIAZHUANG HENRYTE CHEMICALS CO,.LTD(expird)

Contact:+86-311-85208698 311-80837698

Address:NO.166, yuhua west road, SHIJIAZHUANG, China
hangzhou verychem science and technology co.ltd

website:http://www.verypharm.com

Contact:+86-571-88162785; 88162786

Address:F1502, 753 Shenhua road, Hangzhou, China
Zhuhai Rundu Pharmaceutical co.,Ltd

Contact:+86-756-7630755

Address:No.6,North Airport Road,Sanzao Town,Jinwan District

Relevant to this article

Photocatalyzed ortho-Alkylation of Pyridine N-Oxides through Alkene Cleavage

Doi:10.1002/anie.201801305
(2018)
Coordination chemistry of the tetraphenyldithioimidodiphosphinate ligand [Ph₂P(S)NP(S)Ph₂]^? and Ph₂P(CH₂)_nPPh₂, n?=?1, 2, 3 toward ReBr(CO)₅

Doi:10.1016/j.ica.2018.12.024
(2019)
A rapid tandem knoevenagel/michael reaction using mohr's salt as a highly efficient catalyst: Green synthesis of bis(pyrazolyl)methanes

Doi:10.2174/1570178612666141204224826
(2015)
Enantioselective epoxidation of unfunctionalized olefins using chiral (salen)manganese(III) complexes

Doi:10.1016/S0040-4039(00)74486-8
(1991)
Synthesis of sequentially deuterated 1-n-Butyl-3-methylimidazolium ionic liquids

Doi:10.1002/jlcr.1884
(2011)
Optically pure bulky (hetero)arylalkyl carbinols via kinetic resolution

Doi:10.1039/c1cc14591f
(2011)

Article Doi