Bioorganic and Medicinal Chemistry p. 6929 - 6939 (2012)
Update date:2022-09-26
Topics:
Vaidyanathan
White
Affleck
Zhao
Welsh
McDougald
Choi
Zalutsky
A major drawback of internalizing monoclonal antibodies (mAbs) radioiodinated with direct electrophilic approaches is that tumor retention of radioactivity is compromised by the rapid washout of iodo-tyrosine, the primary labeled catabolite for mAbs label
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