
Journal of Medicinal Chemistry p. 3573 - 3578 (1992)
Update date:2022-08-04
Topics:
Naylor, Matthew A.
Threadgill, Michael D.
Webb, Paul
Stratford, Ian J.
Stephens, Miriam A.
et al.
A series of 2-nitroimidazoles bearing side chains terminating in or containing aziridinyl and oxiranyl groups has been prepared, and the compounds were evaluated in vitro as hypoxia-selective bioreductively-activated cytotoxins and selected compounds test
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