Journal of Organic Chemistry p. 5288 - 5294 (2018)
Update date:2022-08-03
Topics:
Li, Yue
Peng, Jinsong
Chen, Xin
Mo, Baichuan
Li, Xue
Sun, Peng
Chen, Chunxia
Multisubstituted indoles were synthesized via a one-pot tandem copper-catalyzed Ullmann-type C-N bond formation/intramolecular cross-dehydrogenative coupling process at 130 °C in DMSO. The methodology allows practical and modular assembly of indoles in go
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