Synthesis of a B-homo 6-azaandrost-4-ene-3-one as a novel steroidal 5α- reductase inhibitor

DOI: 10.1016/S0040-4039(00)76634-2

Source and publish data:

Tetrahedron Letters p. 2823 - 2826 (1994)

Update date:2022-09-26

Topics:

Authors:

Maloney Maloney

Fang Fang

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Article abstract of DOI:10.1016/S0040-4039(00)76634-2

The preparation of a B-ring homologated analog of 17β-N,N- diethylcarboxy-6-azaandrost-4-ene-3-one, a potent inhibitor of type 2 steroidal 5α-reductase, is described.

Full text of DOI:10.1016/S0040-4039(00)76634-2

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