A facile synthesis of 2,3-disubstituted pyrrolo[2,3-b]pyridines via palladium-catalyzed heteroannulation with internal alkynes

DOI: 10.1016/S0040-4039(97)10662-1

Source and publish data:

Tetrahedron Letters p. 627 - 630 (1998)

Update date:2022-08-03

Topics:

Authors:

Park, Sang Sun

Choi, Joong-Kwon

Yum, Eul Kgun

Ha, Deok-Chan

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(97)10662-1

2,3-Disubstituted pyrrolo[2,3-b]pyridines were synthesized by palladium-catalyzed heteroannulation of 2-amino-3-iodopyridine derivatives and internal alkynes with Pd(OAc)₂, LiCl, and KOAc in DMF. The 2-trimethylsilyl-3-methylpyrrolo[2,3-b]pyrid

Full text of DOI:10.1016/S0040-4039(97)10662-1

Products guided by the article

Product name:1-Benzyl-3-methyl-2-trimethylsilanyl-1H-pyrrolo[2,3-b]pyridine

Cas No:203635-50-1

R&D Labs maybe for 203635-50-1

Taizhou Chemedir Biopharm-tech Co., Ltd

Contact:+86 523 86200218

Address:G09, No. 1 Avenue China Medical City, Taizhou,Jiangsu, China
Xi'an caijing Opto-Electrical Science & Technology Co., LTD

Contact:+86-29-88294447

Address:NO.168 Zhangba Rd. East, Xi'an, P.R.China
Exploiter Molybdenum Co.,Ltd

Contact:86-379-63338609

Address:Jiudian Village,Deting Town,Song County,Luoyang
GUANGZHOU MEDCAN PHARMATECH LTD

website:http://www.gzmedcan.com

Contact:+86-20-82519649

Address:Building J,Room 101,1 JiangtashanRd,Guang Zhou Science City,Guang Zhou ,China
Winchem Industrial Co. Ltd.(expird)

Contact:86-574-83851061 86-574-87083208

Address:Room 905, No.3 Building,East Business Center, 456 Xingning Road, Ningbo City,China

Relevant to this article

Enantioselective synthesis of 4-aminocyclopent-2-ene-1-one from tricyclo[5.2.1.0^2,6]decenyl enaminones

Doi:10.1016/S0040-4039(97)10820-6
(1998)
Ionic liquid brush as an efficient and reusable heterogeneous catalytic assembly for the tosylation of phenols and alcohols in neat water

Doi:10.1039/c7nj00141j
(2017)
1,2,4-Triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A₃ adenosine receptor antagonists: Synthesis, pharmacological, and ligand-receptor modeling studies

Doi:10.1021/jm031136l
(2004)
Aryl biphenyl-3-ylmethylpiperazines as 5-HT₇ receptor antagonists

Doi:10.1002/cmdc.201300240
(2013)
Dually acting nonclassical 1,4-dihydropyridines promote the anti-tuberculosis (Tb) activities of clofazimine

Doi:10.3390/molecules24162873
(2019)
Regiochemical Control in the Diels-Alder Reaction of Substituted Naphthoquinones. The Directing Effects of C-6 Oxygen Substituents

Doi:10.1021/jo00146a034
(1982)

Article Doi