
Tetrahedron p. 11907 - 11924 (1998)
Update date:2022-07-29
Topics:
Harburn, James J.
Loftus, Gabrielle C.
Marples, Brian A.
The design and synthesis of potential steroidal HIV-1 protease inhibitors is described. Compounds derived from 1 [-amino-12-keto-cholanic acid derivatives show modest activity.
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