PF1022A - A novel anthelmintic cyclooctadepsipeptide. Modification and exchange of the N-methyl leucine residues

DOI: 10.1016/S0960-894X(98)00156-5

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 1035 - 1040 (1998)

Update date:2022-08-04

Topics:

Authors:

Scherkenbreck, Juergen

Harder, Achim

Plant, Andrew

Dyker, Hubert

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0960-894X(98)00156-5

The first structure-activity relationships of the anthelmintic cyclooctadepsipeptide PF1022A have been established via a systematic exchange of the leucine residues by a series of related N-alkylated amino acids. The data presented strongly suggest that (

Full text of DOI:10.1016/S0960-894X(98)00156-5

Products guided by the article

Product name:L-Leucine, N-methyl-N-(phenylmethyl)-

Cas No:60643-14-3

R&D Labs maybe for 60643-14-3

Daqing New Century Fine Chemical Co., Ltd.(expird)

Contact:010-57126694

Address:No.39, jinxing cun, honggang district
Tianjin Bright Future Technology Co., Ltd

Contact:0086-22-58016666

Address:NO.136 DongTeng Lake Street Tianjin Economic and Technology Development Area,Tainjin,China
Shanghai Dano Pharmaceutical Co.,Ld.(expird)

Contact:+86-592-6266840

Address:Building 1 Room 512, 720 Cailun Rd, Zhangjiang High-Tech Park, Shanghai 201203, China
Chengdu Green Young Biopharmaceutical INC

Contact:+86-28-85337952

Address:1-B-26,Tianhe Industry Park, No.1480 of Tianfu Road,Chengdu,P.R.China,610000
Taizhou Elitechemie MediPharma Technology Co.,Ltd.

Contact:+86-523-86810021

Address:Building G14,NO.1 Avenue,China Medical City, Taizhou, Jiangsu,China

Relevant to this article

Doi:10.1021/ja00432a038
(1976)
AN EFFICIENT SYNTHESIS OF OPTICALLY PURE ANTHRACYCLINONE INTERMEDIATES BY THE NOVEL USE OF MICROBIAL REDUCTION

Doi:10.1016/S0040-4039(00)88665-7
(1982)
High Yielding Acid-Catalysed Hydrolysis of Cellulosic Polysaccharides and Native Biomass into Low Molecular Weight Sugars in Mixed Ionic Liquid Systems

Doi:10.1002/open.201900283
(2019)
A Cu²⁺ protein cavity mimicking fluorescent chemosensor for selective Cu²⁺ recognition: tuning of fluorescence quenching to enhancement through spatial placement of anthracene unit

Doi:10.1016/j.tet.2007.08.101
(2007)
Substituted 6-amino-4H-[1,2]dithiolo[4,3-b]pyrrol-5-ones: Synthesis, structure-activity relationships, and cytotoxic activity on selected human cancer cell lines

Doi:10.1016/j.bmc.2007.04.017
(2007)
Practical synthesis of a highly functionalized thiazole ketone

Doi:10.1016/S0040-4020(03)00878-0
(2003)

Article Doi