Potent and selective antagonists of the antidiuretic responses to arginine-vasopressin based on modifications of [1-(β-mercapto-β,β-pentamethylenepropionic acid),2-D-isoleucine,4-valine]arginine-vasopressin at position 4

Article abstract of DOI:10.1021/jm00370a002

As part of a program in which we are attempting (a) to obtain more potent and/or more selective antagonists of the antidiuretic responses to arginine-vasopressin (AVP) and (b) to delineate the structural features at positions 1-9 required for antidiuretic