The histamine H2 receptor agonist impromidine: Synthesis and structure-activity considerations

DOI: 10.1021/jm00148a007

Source and publish data:

Journal of Medicinal Chemistry p. 1414 - 1422 (1985)

Update date:2022-08-05

Topics:

Authors:

Durant Durant

Ganellin

Hills Hills

et al. et al.

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Article abstract of DOI:10.1021/jm00148a007

Impromidine (1) is a potent and selective histamine H₂ receptor agonist and its structure comprises a strongly basic guanidine group containing two different imidazole-containing side chains. In this paper we report the synthesis of analogues i

Full text of DOI:10.1021/jm00148a007

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