European Journal of Medicinal Chemistry p. 511 - 518 (2018)
Update date:2022-08-28
Topics:
Chernysheva, Natalia B.
Maksimenko, Anna S.
Andreyanov, Fedor A.
Kislyi, Victor P.
Strelenko, Yuri A.
Khrustalev, Victor N.
Semenova, Marina N.
Semenov, Victor V.
4,5-Diarylisoxazoles are potent antiproliferative tubulin-targeting agents. Their isomeric 3,4-diaryl-5-unsubstituted isoxazoles are hardly accessible. The synthesis of 3,4-diaryl-5-unsubstituted isoxazoles 13 was designed based on a condensation of arylb
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