Synthesis of Carbon-14 labeled CI-1012 and CI-1013, potential anti-HIV agents

Article abstract of DOI:10.1002/(SICI)1099-1344(199909)42:9<827::AID-JLCR243>3.0.CO;2-V

¹⁴C-Labeled CI-1012 and CI-1013 of the 2,2'-dithiobis[benzamide] and benzisothiazolone series, inhibitors of viral replication and potential anti-HIV agents, were prepared. The radiolabeling of CI-1013, a six-step synthetic sequence, started wi