Mapping the Melatonin Receptor. 3. Design and Synthesis of Melatonin Agonists and Antagonists Derived from 2-Phenyltryptamines

DOI: 10.1021/jm00007a010

Source and publish data:

Journal of Medicinal Chemistry p. 1132 - 1139 (1995)

Update date:2022-08-30

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Authors:

Garratt, Peter J.

Jones, Rob

Tocher, Derek A.

Sugden, David

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Article abstract of DOI:10.1021/jm00007a010

Three series of 2-phenyltryptamides were prepared as melatonin analogues to investigate the nature of the binding site of the melatonin receptor in chicken brain and in Xenopus laevis melanophore cells.The 5-methoxy-2-phenyltryptamides (6a-j) have high bi

Full text of DOI:10.1021/jm00007a010

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