European Journal of Medicinal Chemistry p. 145 - 155 (2015)
Update date:2022-08-30
Topics:
Yang, Tianming
Chen, Xiao
Jin, Hai-Xiao
Sethi, Gautam
Go, Mei-Lin
Sirtuins are protein deacylases with regulatory roles in metabolism and stress response. Functionalized tetrahydro-1H-pyrido[4,3-b]indoles were identified as preferential sirtuin 2 inhibitors, with in vitro inhibitory potencies in the low micromolar conce
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