4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95%

Base Information

• Chemical Name: 4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95%
• CAS No.: 1239481-05-0
• Molecular Formula: C13H20BN3O3
• Molecular Weight: 259.116
• Hs Code.: 2934999090
• Mol file: 1239481-05-0.mol

Synonyms:4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95%;2-(4-(Azidomethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane

Chemical Property of 4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95%

Chemical Property:

• PSA: 68.21000
• LogP: 2.24886

Purity/Quality:

97% ^*data from raw suppliers

2-(4-(AZIDOMETHYL)PHENYL)-4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLANE ^*data from reagent suppliers

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

SDS file from LookChem

Useful:

Technology Process of 4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95%

There total 3 articles about 4-(AzidoMethyl)benzeneboronic acid pinacol ester, 95% which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 100.0%

C22H29BN2O4S → 2-(4-(azidomethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane (1239481-05-0)

Guidance literature:

In tetrahydrofuran; at 60 ℃; for 0.0833333h;

DOI:10.1246/cl.210204

Reference yield: 99.5%

4-bromomethylphenylboronic acid pinacol ester (138500-85-3) → 2-(4-(azidomethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane (1239481-05-0)

Guidance literature:

With sodium azide; In ethanol; at 20 ℃; for 24h;

DOI:10.1016/j.tetlet.2010.05.104

Reference yield:

4-formylphenylboronic acid, (87199-17-5) → 2-(4-(azidomethyl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane (1239481-05-0)

Guidance literature:

Multi-step reaction with 3 steps

1: methanol / 2 h / 20 °C

2: tetrahydrofuran / 2 h / Reflux

3: tetrahydrofuran / 0.08 h / 60 °C

In tetrahydrofuran; methanol;

DOI:10.1246/cl.210204

upstream raw materials:

4-bromomethylphenylboronic acid pinacol ester

4-formylphenylboronic acid,

Downstream raw materials:

1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)-4-propyl-1,2,3-triazole

4-phenyl-1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)-1H-1,2,3-triazole

2(1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)-1,2,3-triazol-4-yl)propan-2-ol

ethyl 1-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)-1,2,3-triazole-4-carboxylate

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