(2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine

Base Information

• Chemical Name: (2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine
• CAS No.: 107036-26-0
• Molecular Formula: C₂₃H₂₅NO₅
• Molecular Weight: 395.455
• Mol file: 107036-26-0.mol

Synonyms:(2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine

Chemical Property of (2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine

Chemical Property:

Purity/Quality:

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

Useful:

Technology Process of (2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine

There total 1 articles about (2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 98.0%

ethyleneimine (151-56-4,9002-98-6) + Acetic acid 4-[(1S,2R)-2-(4-acetoxy-phenyl)-1-chlorocarbonyl-butyl]-phenyl ester (107036-23-7) → (2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine (107036-26-0)

Guidance literature:

With triethylamine; In diethyl ether; 1.) -4 deg C, 20 min, 2.) RT, 1 h;

DOI:10.1021/jm00388a015

Reference yield: 90.0%

(2R*,3S*)-1-<2,3-bis(4-acetoxyphenyl)-1-pentanoyl>aziridine (107036-26-0) → (2R*,3S*)-1-<2,3-bis(4-hydroxyphenyl)-1-pentanoyl>aziridine (107036-11-3)

Guidance literature:

With potassium carbonate; In methanol; for 1h; Ambient temperature;

DOI:10.1021/jm00388a015

upstream raw materials:

ethyleneimine

Acetic acid 4-[(1S,2R)-2-(4-acetoxy-phenyl)-1-chlorocarbonyl-butyl]-phenyl ester

Downstream raw materials:

(2R*,3S*)-1-<2,3-bis(4-hydroxyphenyl)-1-pentanoyl>aziridine