4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide

Base Information

• Chemical Name: 4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide
• CAS No.: 942263-55-0
• Molecular Formula: C₂₂H₃₀N₂O₃S₂
• Molecular Weight: 434.624

Synonyms:4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide

Chemical Property of 4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide

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Technology Process of 4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide

There total 1 articles about 4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 50.0%

N-(1-[(4-methylphenyl)sulfonyl]tetrahydro-1H-pyrrol-2-yl)-2-methyl-2-propanesulfinamide (918954-35-5) + 1-benzyl-tetrahydro-thiophenium tetrafluoroborate → (Rs,2S,3S)-4-methyl-N-{3-[(2S,3R)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide + 4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide (942263-55-0) + 4-methyl-N-{3-[(2R,3R)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide

Guidance literature:

With phosphoric triamide-based reagent; In tetrahydrofuran; at 0 ℃; for 3.5h;

DOI:10.1021/ol070507f

Reference yield: 93.0%

4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide (942263-55-0) → (R)-2-methylpropane-2-sulfinic acid (2R,3S)-[2-phenyl-1-(toluene-4-sulfonyl)piperidin-3-yl]-amide (942263-58-3)

Guidance literature:

With ytterbium(III) triflate; In dichloromethane; at 20 ℃; for 48h;

DOI:10.1021/ol070507f

Reference yield: 81.0%

4-methyl-N-{3-[(2S,3S)-3-phenyl-1-((R)-2-methylpropane-2-sulfinyl)-aziridin-2-yl]propyl}-benzenesulfonamide (942263-55-0) → (2S,3S)-4-methyl-N-{3-[3-phenylaziridin-2-yl]propyl}-benzenesulfonamide

Guidance literature:

With hydrogenchloride; In 1,4-dioxane; ethanol;

DOI:10.1021/ol070507f

upstream raw materials:

N-(1-[(4-methylphenyl)sulfonyl]tetrahydro-1H-pyrrol-2-yl)-2-methyl-2-propanesulfinamide

Downstream raw materials:

(R)-2-methylpropane-2-sulfinic acid (2R,3S)-[2-phenyl-1-(toluene-4-sulfonyl)piperidin-3-yl]-amide

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