1003319-99-0Relevant articles and documents
Discovery of oxathiapiprolin, a new oomycete fungicide that targets an oxysterol binding protein
Pasteris, Robert J.,Hanagan, Mary Ann,Bisaha, John J.,Finkelstein, Bruce L.,Hoffman, Lisa E.,Gregory, Vann,Andreassi, John L.,Sweigard, James A.,Klyashchitsky, Boris A.,Henry, Yewande T.,Berger, Richard A.
, p. 354 - 361 (2016/01/25)
Oxathiapiprolin is the first member of a new class of piperidinyl thiazole isoxazoline fungicides with exceptional activity against plant diseases caused by oomycete pathogens. It acts via inhibition of a novel fungal target - an oxysterol binding protein - resulting in excellent preventative, curative and residual efficacy against key diseases of grapes, potatoes and vegetables. Oxathiapiprolin is being developed globally as DuPont Zorvec disease control with first registration and sales anticipated in 2015. The discovery, synthesis, optimization and biological efficacy are presented.
Piperidinyl thiazole isoxazolines: A new series of highly potent, slowly reversible FAAH inhibitors with analgesic properties
Pember, Stephen O.,Mejia, Galo L.,Price, Theodore J.,Pasteris, Robert J.
, p. 2965 - 2973 (2016/06/06)
Fatty acid amide hydrolase (FAAH) is a membrane anchored serine hydrolase that has a principle role in the metabolism of the endogenous cannabinoid anandamide. Docking studies using representative FAAH crystal structures revealed that compounds containing
AZOCYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE
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Page/Page column 47, (2011/06/26)
Disclosed are compounds of Formula 1, including all stereoisomers, N oxides, and salts thereof, wherein A, W, X, G, R1, R2, R3, R4, m and n are as defined in the disclosure. Also disclosed are pharmaceutical compositions containing the compounds of Formula 1 and methods for treating a disease or condition mediated by fatty acid amide hydrolase activity comprising applying a therapeutically effective amount of a compound or a composition of the invention
FUNGICIDAL MIXTURES
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Page/Page column 58, (2010/10/03)
Disclosed is a fungicidal composition comprising (a) at least one compound selected from the compounds of Formula 1 N-oxides, and salts thereof, wherein R1, R2, A, G, W, Z1, X, J, and n are as defined in the disclosure, and (b) at least one additional fungicidal compound. Also disclosed is a method for controlling plant diseases caused by fungal plant pathogens comprising applying to the plant or portion thereof, or to the plant seed, a fungicidally effective amount of the aforesaid composition. Also disclosed is a composition comprising component (a) of aforesaid composition and at least one insecticide. Also disclosed are compounds of Formula 1A, 1B and 1C, wherein R1, R2, A, G, W, Z1, X, J, n, Z3, M and J1 are as defined in the disclosure.
FUNGICIDAL HETERCYCLIC COMPOUNDS
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Page/Page column 129, (2009/09/05)
Disclosed are compounds of Formula (1), including all geometric and stereoisomers, N-oxides, and salts thereof, formula (1) wherein E, R2, G, Z1, J and n are as defined in the disclosure. Also disclosed are compositions containing th
ELECTRONIC COMPONENT HAVING FLEXIBLE PRINTED CIRCUIT BOARD TECHNOLOGY
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Page/Page column 75, (2008/06/13)
The invention relates to an electronic component (1) having a housing comprising at least one base plate (3), a housing cover, and at least two electronic connections (5) between substrates (7) disposed in the interior of the housing and components located outside the housing in the form of printed circuit boards, which can be at least partially fixed on the base plate (3), wherein at least one first partially flexible printed circuit board (5a) and a second printed circuit board (5b) are configured such that they overlap at least in one region (6) in the assembled state. The invention further relates to a method for the production of such an electronic component.